Is a
Patent attributes
Patent Jurisdiction
Patent Number
Patent Inventor Names
Maria E. Gaczynska0
Pawel A. Osmulski0
Date of Patent
January 1, 2019
Patent Application Number
14896984
Date Filed
June 13, 2014
Patent Citations Received
Patent Primary Examiner
Patent abstract
The present invention relates generally to novel allosteric regulators of proteasome activity, methods for preparation and use, and pharmaceutical compositions thereof. Specifically piperidine-2-carboxylic acid derivatives containing 1-oxo-aroyl group and a lipophilic ester side chain are disclosed as allosteric inhibitors of proteasome 2S activity, and as therapeutic agents for the treatment of proteasome-associated disorders in a subject.
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