Is a
Patent attributes
Patent Applicant
Current Assignee
Patent Jurisdiction
Patent Number
Patent Inventor Names
Theresa Cravillion0
Qingping Tian0
Stephan Bachmann0
Sushant Malhotra0
Alec Fettes0
Alexander Gmehling0
Danial Beaudry0
Francis Gosselin0
...
Date of Patent
August 20, 2019
Patent Application Number
15841828
Date Filed
December 14, 2017
Patent Citations Received
Patent Primary Examiner
Patent abstract
Methods for preparing the Bruton's Tyrosine Kinase (“BTK”) inhibitor compound 2-{3′-hydroxymethyl-1-methyl-5-[5-((S)-2-methyl-4-oxetan-3-yl-piperazin-1-yl)-pyridin-2-ylamino]-6-oxo-1,6-dihydro-[3,4′]bipyridinyl-2′-yl}-7,7-dimethyl-3,4,7,8-tetrahydro-2H,6H-cyclopenta[4,5]pyrrolo[1,2-a]pyrazin-1-one are provided. Methods for preparing tricyclic lactam compounds are also provided.
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