Is a
Patent attributes
Current Assignee
Patent Jurisdiction
Patent Number
Patent Inventor Names
John C. Prescott0
Andrew Braisted0
Date of Patent
April 10, 2007
0Patent Application Number
103943220
Date Filed
March 20, 2003
0Patent Primary Examiner
Patent abstract
The invention concerns the identification of protein kinase inhibitors that preferentially bind to the inactive conformation of a target protein kinase. The inhibitors are identified by locking the target protein kinase in an inactive conformation, and using a covalent tethering approach to identify inhibitors preferentially targeting the inactive conformation.
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