Is a
Patent attributes
Patent Jurisdiction
Patent Number
Date of Patent
January 29, 2008
Patent Application Number
11233845
Date Filed
September 21, 2005
Patent Primary Examiner
Patent abstract
This invention relates to a new and convergent route to small molecule inhibitors of poly(ADP-ribose) polymerase, such as 8-fluoro-2-{4-[(methylamino)methyl]phenyl}-1,3,4,5-tetrahydro-6H-azepino[5,4,3-cd]indol-6-one, via a key Sonogashira coupling reaction and a CuI-promoted indole formation.
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